发明名称 |
Notkun ß esterum af L-karnitÝni e-a alkan¾²l L-karnitÝni sem katj¾nÝsk lÝpÝ- fyrir innanfrumu dreifinguna ß lyfjafrµ-ilega virkum efnasamb÷ndum |
摘要 |
The use of esters of L-carnitine and alkanoyl L-carnitines as cationic lipids for the intracellular delivery of pharmacologically active compounds is described. The esters according to the invention have general formula (II) <CHEM> wherein the R groups are as defined in the description. |
申请公布号 |
IS8719(A) |
申请公布日期 |
2008.03.07 |
申请号 |
IS20080008719 |
申请日期 |
2008.03.07 |
申请人 |
SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. |
发明人 |
CLAUDIO PISANO;MARIA ORNELLA TINTI;MOSE SANTANIELLO;LUCIANA CRITELLI |
分类号 |
A61K8/00;A61K8/11;A61K8/14;A61K8/30;A61K8/37;A61K8/44;A61K9/127;A61K31/225;A61K31/337;A61K31/4745;A61K39/00;A61K45/00;A61K47/18;A61K47/24;A61K47/44;A61K48/00;A61P35/00;A61Q19/00;C07C229/02;C07C229/22 |
主分类号 |
A61K8/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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