发明名称 KV1.5 POTASSIUM CHANNEL INHIBITORS
摘要 The present invention relates to 4-oxo-1,3,8-triaza-spiro[4.5]decanes which are useful as Kv1.5 potassium channel inhibitors providing atrial-selective antiarrhythmic activity. The present invention further relates to compositions and methods for treating atrial-selective antiarrhythmia.
申请公布号 WO2007149873(A3) 申请公布日期 2008.03.06
申请号 WO2007US71586 申请日期 2007.06.19
申请人 WYETH;JANUSZ, JOHN, MICHAEL;WU, SHENGDE;FAIRWEATHER, NEIL, T.;LEE, WENLIN;BLASS, BENJAMIN, E.;FLUXE, ANDREW, J.;HODSON, STEPHEN, J.;RIDGEWAY, JAMES, M, II 发明人 JANUSZ, JOHN, MICHAEL;WU, SHENGDE;FAIRWEATHER, NEIL, T.;LEE, WENLIN;BLASS, BENJAMIN, E.;FLUXE, ANDREW, J.;HODSON, STEPHEN, J.;RIDGEWAY, JAMES, M, II
分类号 C07D471/10;A61K31/505;A61P9/06 主分类号 C07D471/10
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