发明名称 POLYMORPH OF (R) -3- (2-HYDROXY-2, 2-DIPHENYL-ACETOXY) -1- (ISOXAZOL-3-YLCARBAMOYL-METHYL) -1-AZONI A-BICYCLO- [2.2.2] OCTANE BROMIDE
摘要 A novel polymorphic crystal form of (R)-3-(2-hydroxy-2,2-diphenyl-acetoxy )-1-(isoxazol-3- ylcarbamoyl-methyl)-1-azonia-bicyclo-[2.2.2]octane bromide, designated crystal form Talpha. Methods for preparing same and the use of t he crystal form as the active ingredient of medicaments for the treatment of inflammatory or obstructive airways diseases are also described.
申请公布号 CA2660983(A1) 申请公布日期 2008.03.06
申请号 CA20072660983 申请日期 2007.08.29
申请人 NOVARTIS AG 发明人 MUHRER, GERHARD;MONNIER, STEPHANIE
分类号 C07D453/02;A61K31/439;A61P11/06 主分类号 C07D453/02
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