发明名称 QUINAZOLINES FOR PDK1 INHIBITION
摘要 The invention provides quinazoline compounds that are inhibitors of PDKl. Also provided are pharmaceutical compositions including the compounds, and methods of treating proliferative diseases, such as cancers, with the compounds or compositions.
申请公布号 WO2007117607(A9) 申请公布日期 2008.03.06
申请号 WO2007US08592 申请日期 2007.04.05
申请人 NOVARTIS VACCINES & DIAGNOSTICS, INC.;RAMURTHY, SAVITHRI;LIN, XIADONG;SUBRAMANIAN, SHARADA;RICO, ALICE, C.;WANG, XIAJONG, M.;JAIN, RAMA;MURRAY, JEREMY, M.;BASMAN, STEVEN, E.;WARNE, ROBERT, L.;SHU, WEI;ZHOU, YASHEEN;DOVE, JEFFREY;AIKAWA, MINA;AMIRI, PAYMAN;WANG, WEIBO;JANSEN, JOHANNA, M.;WAGMAN, ALLAN, S.;PFISTER, KEITH, B.;NG, SIMON, C. 发明人 RAMURTHY, SAVITHRI;LIN, XIADONG;SUBRAMANIAN, SHARADA;RICO, ALICE, C.;WANG, XIAJONG, M.;JAIN, RAMA;MURRAY, JEREMY, M.;BASMAN, STEVEN, E.;WARNE, ROBERT, L.;SHU, WEI;ZHOU, YASHEEN;DOVE, JEFFREY;AIKAWA, MINA;AMIRI, PAYMAN;WANG, WEIBO;JANSEN, JOHANNA, M.;WAGMAN, ALLAN, S.;PFISTER, KEITH, B.;NG, SIMON, C.
分类号 C07D239/94;C07D401/04;C07D401/06;C07D401/12;C07D401/14;C07D403/04;C07D403/06;C07D403/10;C07D403/12;C07D403/14;C07D405/04;C07D405/12;C07D405/14;C07D409/12;C07D413/04;C07D413/12 主分类号 C07D239/94
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