发明名称 METHOD FOR PRODUCING PHENOXYPYRIDINE DERIVATIVE
摘要 <p>Disclosed is a method for producing a compound represented by the formula (I) below, which is characterized in that a compound represented by the formula (II) below or a salt thereof is reacted with a compound represented by the formula (III) below in the presence of a condensing agent. (II) [In the formula, R&lt;SUP&gt;1&lt;/SUP&gt; represents (1) an optionally substituted acetidin-1-yl group, (2) an optionally substituted pyrrolidin-1-yl group, (3) an optionally substituted piperidin-1-yl group or the like; and R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, R&lt;SUP&gt;4&lt;/SUP&gt; and R&lt;SUP&gt;5&lt;/SUP&gt; may be the same or different and represent a hydrogen atom or afluorine atom.] (III) [In the formula, R&lt;SUP&gt;6&lt;/SUP&gt; represents a hydrogen atom or a fluorine atom.] (I) [In the formula, R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, R&lt;SUP&gt;4&lt;/SUP&gt;, R&lt;SUP&gt;5&lt;/SUP&gt; and R&lt;SUP&gt;6&lt;/SUP&gt; are as defined above.]</p>
申请公布号 WO2008026577(A1) 申请公布日期 2008.03.06
申请号 WO2007JP66635 申请日期 2007.08.28
申请人 EISAI R & D MANAGEMENT CO., LTD.;NAGAI, MITSUO;MATSUSHIMA, TOMOHIRO;KAMADA, ATSUSHI;WAKASUGI, KAZUNORI;SHIROTORI, SHUJI;ABE, SHINYA;NARA, KAZUMASA;SAKAGUCHI, TAKAHISA 发明人 NAGAI, MITSUO;MATSUSHIMA, TOMOHIRO;KAMADA, ATSUSHI;WAKASUGI, KAZUNORI;SHIROTORI, SHUJI;ABE, SHINYA;NARA, KAZUMASA;SAKAGUCHI, TAKAHISA
分类号 C07D213/73;A61K31/4427;A61K31/4439;A61K31/4545;A61K31/496;A61P9/00;A61P35/00;A61P35/04;A61P43/00;C07D213/75;C07D213/81;C07D401/12 主分类号 C07D213/73
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