发明名称 NOVEL MCH RECEPTOR ANTAGONISTS
摘要 The present invention relates to a melanin concentrating hormone antagonist compound of formula (I): wherein R<SUP>1</SUP>, R<SUP>a</SUP>, R<SUP>b</SUP>, R<SUP>2</SUP>, L<SUP>1</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP> and R<SUP>5</SUP> are as defined, or a pharmaceutically acceptable salt, enantiomer, diastereomer or mixture of diastereomers thereof useful in the treatment, obesity and related diseases.
申请公布号 WO2007146759(A3) 申请公布日期 2008.02.21
申请号 WO2007US70668 申请日期 2007.06.08
申请人 ELI LILLY AND COMPANY;AMEGADZIE, ALBERT, KUDZOVI;DAO, YEN;GARDINIER, KEVIN, MATTHEW;GARMENE, DAVID, JOSEPH;GREEN, STEVEN, JAMES;HEMBRE, ERIK, JAMES;LU, JIANLIANG;SPINAZZE, PATRICK, GIANPIETRO 发明人 AMEGADZIE, ALBERT, KUDZOVI;DAO, YEN;GARDINIER, KEVIN, MATTHEW;GARMENE, DAVID, JOSEPH;GREEN, STEVEN, JAMES;HEMBRE, ERIK, JAMES;LU, JIANLIANG;SPINAZZE, PATRICK, GIANPIETRO
分类号 C07D495/04;A61K31/4365;A61P3/04 主分类号 C07D495/04
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