摘要 |
The present invention relates to a melanin concentrating hormone antagonist compound of formula (I): wherein R<SUP>1</SUP>, R<SUP>a</SUP>, R<SUP>b</SUP>, R<SUP>2</SUP>, L<SUP>1</SUP>, R<SUP>3</SUP>, R<SUP>4</SUP> and R<SUP>5</SUP> are as defined, or a pharmaceutically acceptable salt, enantiomer, diastereomer or mixture of diastereomers thereof useful in the treatment, obesity and related diseases. |
申请人 |
ELI LILLY AND COMPANY;AMEGADZIE, ALBERT, KUDZOVI;DAO, YEN;GARDINIER, KEVIN, MATTHEW;GARMENE, DAVID, JOSEPH;GREEN, STEVEN, JAMES;HEMBRE, ERIK, JAMES;LU, JIANLIANG;SPINAZZE, PATRICK, GIANPIETRO |
发明人 |
AMEGADZIE, ALBERT, KUDZOVI;DAO, YEN;GARDINIER, KEVIN, MATTHEW;GARMENE, DAVID, JOSEPH;GREEN, STEVEN, JAMES;HEMBRE, ERIK, JAMES;LU, JIANLIANG;SPINAZZE, PATRICK, GIANPIETRO |