| 发明名称 |
Process for cross coupling indoles |
| 摘要 |
The present invention provides a process for making a compound of general formula I: wherein: R=H or C<SUB>1-8</SUB>alkyl X=C<SUB>3</SUB>-C<SUB>8</SUB>cycloalkyl, C<SUB>3</SUB>-C<SUB>8</SUB>aryl or C<SUB>3</SUB>-C<SUB>8</SUB>alkyl; Y=heteroaryl or aryl; Z=H, HO<SUB>2</SUB>C-, C<SUB>1-8</SUB>alkyl O<SUB>2</SUB>C-, C<SUB>1-6</SUB>alkyl HNC(O)-, and as described herein.
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| 申请公布号 |
US7332614(B2) |
申请公布日期 |
2008.02.19 |
| 申请号 |
US20050074194 |
申请日期 |
2005.03.07 |
| 申请人 |
BOEHRINGER INGELHEIM INTERNATIONAL, GMBH |
发明人 |
KHODABOCUS AHMAD;LI GUISHENG;LU ZHI-HUI;ROSCHANGAR FRANK;SENANAYAKE CHRIS HUGH;SHEN MING |
| 分类号 |
C07D209/10;A61K31/404;C07D209/30;C07D417/02 |
主分类号 |
C07D209/10 |
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