摘要 |
PROBLEM TO BE SOLVED: To provide a method for producing a perindopril with the need of neither use of any protecting group nor the step of separating the stereoisomer. SOLUTION: The method for producing a perindopril of the formula(I)(wherein, Ra is H or a 1-4C alkyl; Rb is a 1-4C alkyl; Rc is a 1-9C alkyl; and Rd is H or a protecting group) or a derivative thereof comprises carrying out a reaction between a compound(IV) and a compound(V). COPYRIGHT: (C)2008,JPO&INPIT
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