发明名称 2-Phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
摘要 The present invention relates to new 2-Phenyl-1-[4-(2-Aminoethoxy)-Benzyl]-Indole compounds having the general structures below: which are useful in contraception and in treating melanoma, osteoporosis, acne, dysfunctional uterine bleeding, endometrial polyps, benign breast disease, adenomyosis, infertility, endometriosis, endometrial cancer, polycystic ovary syndrome, cardiovascular disease, Alzheimer's disease, cognitive decline, central nervous system disorders, central nervous system cancers, leukemia, endometrial ablations, chronic renal disease, chronic hepatic disease, coagulation diseases and disorders, hypocalcemia, hypercalcemia, Paget's disease, osteomalacia, osteohalisteresis, and multiple myeloma.
申请公布号 US2008021017(A1) 申请公布日期 2008.01.24
申请号 US20070820735 申请日期 2007.06.20
申请人 WYETH 发明人 MILLER CHRIS P.;COLLINI MICHAEL D.;TRAN BACH D.;SANTILLI ARTHUR A.
分类号 A61K31/404;A61K31/4523;A61K31/496;A61K31/55;A61P3/06;A61P5/00;A61P5/30;A61P9/00;A61P13/08;A61P15/00;A61P17/10;A61P19/10;A61P25/28;A61P35/00;C07D209/08;C07D209/10;C07D209/12;C07D209/30;C07D209/42;C07D403/12;C07D405/04;C07D405/12 主分类号 A61K31/404
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