发明名称 TETRAHYDRO ISOQUINOLINE DERIVATIVES, PREPARATION METHODS AND MEDICINAL USES THEREOF
摘要 <p>A kind of tetrahydro isoquinoline derivatives (I), their preparation methods, medicine compositions and medicinal uses thereof, especially their uses as ?-opioid receptor excitant in pain relieving, which belongs to the medicine chemistry. The subsutituents R&lt;SUP&gt;1&lt;/SUP&gt;,R&lt;SUP&gt;2&lt;/SUP&gt;,R&lt;SUP&gt;3&lt;/SUP&gt;,R&lt;SUP&gt;4&lt;/SUP&gt; of general formula (I) are defined as the description.</p>
申请公布号 WO2008009215(A1) 申请公布日期 2008.01.24
申请号 WO2007CN02115 申请日期 2007.07.10
申请人 CHINA PHARMACEUTICAL UNIVERSITY;SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES;XU, YUNGEN;LIU, JINGGEN;GUO, TING;WANG, DECHUAN 发明人 XU, YUNGEN;LIU, JINGGEN;GUO, TING;WANG, DECHUAN
分类号 C07D217/06;A61K31/472;A61K31/4725;A61P9/12;A61P25/04;A61P25/20;A61P25/36;A61P29/00;A61P31/18;C07D401/06;C07D403/06;C07D471/10 主分类号 C07D217/06
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