发明名称 TARTRATE SALT OF (7S)-7-[(5-FLUORO-2-METHYL-BENZYL)OXY]-2-[(2R)-2-METHYLPIPERAZIN-1-YL]-6,7-DIHYDRO-5H-CYCLOPENTA[B]PYRIDINE
摘要 <p>The present invention provides a tartrate salt of Formula (I), Formula I is also known as (7S)-7-[(5-fluoro-2-methyl-benzyl)oxy]-2-[(2R)-2- methylpiperazin -1-yl]-6,7-dihydro -5H-cyclopenta[b]pyridine. The tartrate salt is preferably crystalline. The tartrate salt of Formula I of the invention is useful in the treatment of diseases linked to activation of the 5HT2c receptor in animals including humans, for example, in the treatment of schizophrenia, cognitive deficits including cognitive deficits associated with schizophrenia, anxiety, depression, obsessive-compulsive disorder, epilepsy, obesity, sexual dysfunction, and urinary incontinence, among others.</p>
申请公布号 WO2008010073(A1) 申请公布日期 2008.01.24
申请号 WO2007IB02025 申请日期 2007.07.09
申请人 PFIZER PRODUCTS INC.;LIU, KEVIN KUN-CHIN;ZENG, YUAN 发明人 LIU, KEVIN KUN-CHIN;ZENG, YUAN
分类号 C07D221/04;A61K31/496;A61P25/00 主分类号 C07D221/04
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