发明名称 PROCESS FOR PRODUCTION OF 1-(3-(2-(1-BENZOTHIOPHEN-5-YL)-ETHOXY)PROPYL)AZETIDIN-3-OL OR SALTS THEREOF
摘要 A process for the production of 1-(3-(2-(1-benzothiophen-5-yl)ethoxy) propyl)azetidin-3-ol or salts thereof which comprises using as a starting compound a (phenylthio)acetic acid derivative represented by the general formula [1] or a salt thereof: [Chemical Formula 1] (wherein X1 is halogeno) is useful as a safe process for mass production of 1-(3-(2-(1-benzothiophen-5-yl)ethoxy)propyl)azetidin-3-ol or salts thereof which are useful as remedies for central nervous system diseases and peripheral nerve diseases.
申请公布号 KR20080008334(A) 申请公布日期 2008.01.23
申请号 KR20077024039 申请日期 2006.03.27
申请人 TOYAMA CHEMICAL CO., LTD. 发明人 SAITOH AKIHITO;SUZUKI YOSHIAKI;YONEZAWA KENJI;KAWAMURA MITSUHIDE;KUSANAGI TAKAHIKO;NAKAI TAKASHI
分类号 C07D409/12;C07D333/54;C07D333/64 主分类号 C07D409/12
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