发明名称 |
PROCESS FOR PREPARING GABAPENTIN |
摘要 |
A process for preparing gabapentin of formula 1, which comprises Formula (I) converting 1-allyl-cyclohexanecarboxaldehyde into 1-allyl-cyclohexanecar bonitrile; ozonizing 1-allyl-cyclohexanecarbonitrile to obtain 1-cyano-cyclo hexaneacetaldehyde; acetalizing 1-cyano-cyclohexaneacetaldehyde with a suita ble acetalizing agent to give the corresponding acetal and converting the la tter into gabapentin.
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申请公布号 |
CA2660769(A1) |
申请公布日期 |
2008.01.10 |
申请号 |
CA20072660769 |
申请日期 |
2007.06.29 |
申请人 |
ZACH SYSTEM S.P.A. |
发明人 |
GHELFI, FRANCO;COTARCA, LIVIUS;GIOVANETTI, ROBERTO;NICOLI, ANDREA;RONCAGLIA, FABRIZIO |
分类号 |
C07C217/44;C07C227/18;C07C229/28;C07C253/30;C07C255/46;C07D317/28;C07D317/30 |
主分类号 |
C07C217/44 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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