发明名称 PROCESS FOR THE PREPARATION OF ASENAPINE AND INTERMEDIATE PRODUCTS USED IN SAID PROCESS.
摘要 <p>The invention relates to a novel process for the preparation of asenapine, i.e. trans-5- chloro-2-methyl-2,3,3a, 12b-tetrahydro-1 H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole, as well as to novel intermediate products for use in said process.</p>
申请公布号 WO2008003460(A1) 申请公布日期 2008.01.10
申请号 WO2007EP05876 申请日期 2007.07.03
申请人 N.V. ORGANON;KEMPERMAN, GERARDUS, JOHANNES;STUK, TIMOTHY, LEE;LINDEN, VAN DER, JACOBUS, JOHANNES, MARIA 发明人 KEMPERMAN, GERARDUS, JOHANNES;STUK, TIMOTHY, LEE;LINDEN, VAN DER, JACOBUS, JOHANNES, MARIA
分类号 C07D491/04;C07C39/21;C07C69/017;C07D207/08;C07F7/10 主分类号 C07D491/04
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