| 摘要 |
FIELD: organic chemistry, medicine, pharmacy. ^ SUBSTANCE: invention describes compound of the formula (I): or its pharmaceutically acceptable salt or a prodrug of the formula (I) wherein m = 0-2; X means carbon or nitrogen atom; Y means radical of the formula (i) (ii) or each R1 means independently halogen atom, alkyl, alkoxy-group; A means -SO2- or -(C=O)-; R2 means alkyl or -(CH2)p-NRcRd wherein p = 0; each Rc and Rd means independently hydrogen atom or alkyl; each R3, R4, R5 and R6 means independently hydrogen atom or alkyl, and a pharmaceutical composition based on thereof. Represented compounds possess agonistic activity with respect to alpha-1-A/L-adrenergic receptors. ^ EFFECT: valuable medicinal properties of compounds and pharmaceutical composition. ^ 7 cl, 1 tbl, 12 ex |
