发明名称 |
ENANTIOMERS OF N,N-DIMETHYL-3-(2-THIENYL)-3-HYDROXYPROPANAMINE BORANE AS INTERMEDIATES IN THE SYNTHESIS OF DULOXETINE |
摘要 |
Duloxetine intermediates of formulae (I) and (II), processes for their preparation, and their conversion to pharmaceutically acceptable salts of duloxetine are described. |
申请公布号 |
WO2007123900(A3) |
申请公布日期 |
2007.12.21 |
申请号 |
WO2007US09363 |
申请日期 |
2007.04.17 |
申请人 |
TEVA PHARMACEUTICAL INDUSTRIES LTD.;TEVA PHARMACEUTICALS USA, INC;INI, SANTIAGO;SHMUELY, YARON |
发明人 |
INI, SANTIAGO;SHMUELY, YARON |
分类号 |
C07D333/16;C07C29/136;C07F5/02 |
主分类号 |
C07D333/16 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|