发明名称 |
METHOD OF PREPARING 4-HALOGENATED QUINOLINE INTERMEDIATES |
摘要 |
This invention is directed to methods of preparing compounds of formula (I): comprising the step of reacting a compound of formula (II): with a reagent of formula POX<SUB>3</SUB> and silica gel at a temperature greater than about 75°C, and wherein substitutions at X, PG, A, G, R<SUB>1</SUB> and R<SUB>4</SUB> are set forth in the specification. |
申请公布号 |
WO2007139797(A2) |
申请公布日期 |
2007.12.06 |
申请号 |
WO2007US12211 |
申请日期 |
2007.05.23 |
申请人 |
WYETH;BERNIER, CAROLINE;SHAW, CHIA-CHENG |
发明人 |
BERNIER, CAROLINE;SHAW, CHIA-CHENG |
分类号 |
C07D215/56;C07D401/12 |
主分类号 |
C07D215/56 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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