发明名称 |
HETEROCYCLIC COMPOUNDS AS CALCIUM CHANNEL BLOCKERS |
摘要 |
<p>Methods and compounds effective in ameliorating conditions characterized by unwanted calcium channel activity, particularly unwanted N-type calcium channel activity are disclosed. Specifically, a series of heterocyclic compounds are disclosed of the general formula (1) where X<SUP>1</SUP> and X<SUP>2 </SUP>are linkers and W is an optionally substituted imidazolyl, oxazolyl, thiazolyl, benzimidazolyl, benzoxazolyl, or benzothiazolyl.</p> |
申请公布号 |
WO2007137417(A1) |
申请公布日期 |
2007.12.06 |
申请号 |
WO2007CA00943 |
申请日期 |
2007.05.25 |
申请人 |
NEUROMED PHARMACEUTICALS LTD.;PAJOUHESH, HASSAN;DING, YANBING |
发明人 |
PAJOUHESH, HASSAN;DING, YANBING |
分类号 |
C07D417/12;A61K31/496;A61P3/14;C07D403/12;C07D413/12 |
主分类号 |
C07D417/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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