发明名称 PYRIMIDINE COMPOUND CRYSTAL OR AMORPHOUS FORM AND PROCESS FOR PRODUCING THE SAME
摘要 <p>Crystals of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1 H )-one having a diffraction peak at a diffraction angle (2¸ ± 0.2°) of 9.7° and/or 21.9° in a powder X-ray diffraction are suitable for an active ingredient of a preventing and therapeutic agent for diseases such as constipation. Crystals of 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1 H )-one hydrate and amorphous 5-[2-amino-4-(2-furyl)pyrimidin-5-yl]-1-methylpyridin-2(1 H )-one hydrate are also suitable for an active ingredient of a preventing and therapeutic agent for diseases such as constipation.</p>
申请公布号 EP1862463(A1) 申请公布日期 2007.12.05
申请号 EP20060729533 申请日期 2006.03.20
申请人 EISAI R&D MANAGEMENT CO., LTD. 发明人 HARADA, HITOSHI;ISHIHARA, HIROSHI;SATO, YOSHIAKI;CHIBA, HIROYUKI;KOMATSU, YUKI;INOUE, SUSUMU;OZEKI, NAOKI
分类号 C07D405/14;A61K31/506;A61P1/10;C07D405/06 主分类号 C07D405/14
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