发明名称 INDOLE DERIVATIVES AND THEIR USE AS THYROID RECEPTOR LIGANDS
摘要 <p>The invention provides compounds of formula (I) or pharmaceutically acceptable esters, amides, solvates or salts thereof, including salts of such esters or amides, and solvates of such esters, amides or salts, (I) wherein R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, R&lt;SUP&gt;4&lt;/SUP&gt;, R&lt;SUP&gt;5&lt;/SUP&gt;, R&lt;SUP&gt;6&lt;/SUP&gt;, Y and W are as defined in the specification. The invention also provides the use of such compounds in the treatment or prophylaxis of a condition that may be treated with a thyroid receptor agonist or partial agonist.</p>
申请公布号 WO2007134864(A1) 申请公布日期 2007.11.29
申请号 WO2007EP04623 申请日期 2007.05.24
申请人 KARO BIO AB;GARCIA COLLAZO, ANA MARIA;KOCH, EVA, KRISTINA;MALM, LARS, JOHAN;CHENG, AIPING;HANSSON, TOMAS, FREDRIK 发明人 GARCIA COLLAZO, ANA MARIA;KOCH, EVA, KRISTINA;MALM, LARS, JOHAN;CHENG, AIPING;HANSSON, TOMAS, FREDRIK
分类号 C07D209/08;A61K31/404;A61P5/14;C07D209/18;C07D209/20;C07D405/04;C07D413/04 主分类号 C07D209/08
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