发明名称 |
Thiazolo-pyrimidine/pyridine urea derivatives |
摘要 |
There are presented compounds of the formula or a pharmaceutically acceptable salt thereof, which are active adenosine A2B receptor antagonists and useful in the treatment of diabetes, diabetic retinopathy, asthma and diarrhea.
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申请公布号 |
US2007270433(A1) |
申请公布日期 |
2007.11.22 |
申请号 |
US20070801972 |
申请日期 |
2007.05.11 |
申请人 |
BRINKMAN JOHN A;CHEUNG ADRIAN WAI-HING;FIROOZNIA FARIBORZ;GUERTIN KEVIN RICHARD;MARCOPULOS NICHOLAS;QI LIDA;RACHA JAGDISH KUMAR;SARABU RAMAKANTH;TAN JENNY;TILLEY JEFFERSON WRIGHT |
发明人 |
BRINKMAN JOHN A.;CHEUNG ADRIAN WAI-HING;FIROOZNIA FARIBORZ;GUERTIN KEVIN RICHARD;MARCOPULOS NICHOLAS;QI LIDA;RACHA JAGDISH KUMAR;SARABU RAMAKANTH;TAN JENNY;TILLEY JEFFERSON WRIGHT |
分类号 |
A61K31/519;A61K31/496;C07D498/02 |
主分类号 |
A61K31/519 |
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