发明名称 8-(3-AMINO-PIPERIDIN-1-YL)-XANTHINES, THE PRODUCTION THEREOF AND THE USE OF THE SAME AS MEDICAMENTS
摘要 The invention relates to substituted xanthines of general formula (I) wherein R1 to R3 have the designations cited in patent claims 1 to 16, and to the tautomers, stereoisomers, mixtures, prodrugs and salts thereof, which have precious pharmacological properties, especially an inhibiting effect on the activity of the enzyme dipeptidylpeptidase-IV (DPP-IV).
申请公布号 RS20050137(A) 申请公布日期 2007.11.15
申请号 YU2005P000137 申请日期 2003.08.18
申请人 BOEHRINGER INGELHEIM PHARMA GMBH & CO.KG 发明人 HIMMELSBACH FRANK;LANGKOPF ELKE;ECKHARDT MATTHIAS;MARK MICHAEL;MAIER ROLAND;LOTZ RALF RICHARD HERMAN;TADAYYON MOHAMMAD
分类号 C07D473/04;A61K9/02;A61K9/20;A61K9/28;A61K9/48;A61K31/522;A61K47/02;A61P3/10;C07D473/06;C07D473/08 主分类号 C07D473/04
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