发明名称 4- (2, E-DICHLORO-BENZOYLAMINO) -1H-PYRAZOLE-S-CARBOXYLIC ACID (1-METHANESULPH0NYL-PIPERIDIN-4-YL) -AMIDE FOR THE TREATMENT OF CANCER
摘要 <p>The invention provides the compound of formula (I) 4-(2,6-dichloro-benzoylamino)-1H-pyrazole- 3-carboxylic acid (l-methanesulphonyl-piperidin-4-yl)-amide in a substantially crystalline form, therapeutic uses thereof and pharmaceutical compositions containing the crystalline compound. The invention also provides novel pharmaceutical formulations containing 4-(2,6-dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid (1-methanesulphonyl-piperidin-4-yl)-amide and novel processes for preparing the compound.</p>
申请公布号 WO2007129066(A1) 申请公布日期 2007.11.15
申请号 WO2007GB01655 申请日期 2007.05.04
申请人 ASTEX THERAPEUTICS LIMITED;TREWARTHA, GARY;NAVARRO, EVA, FIGUEROA;REES, DAVID, CHARLES;VINKOVIC, MLADEN;WOODHEAD, ANDREW, JAMES;WYATT, PAUL, GRAHAM 发明人 TREWARTHA, GARY;NAVARRO, EVA, FIGUEROA;REES, DAVID, CHARLES;VINKOVIC, MLADEN;WOODHEAD, ANDREW, JAMES;WYATT, PAUL, GRAHAM
分类号 C07D401/12;A61K31/4155;A61P35/00 主分类号 C07D401/12
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