发明名称 NOVEL 3-ARYL-1,2-BENZISOXAZOLE DERIVATIVES, COMPOSITIONS CONTAINING SAME AND USE THEREOF.
摘要 <p>The invention concerns novel products of formula (I), wherein: A1 and A2 represent CH or N; X represents Cra or N; Y represents CRb or N; R<sub>1</sub>, R<sub>2</sub>, R<sub>3</sub> and R<sub>4</sub> identical or different represent in particular hydrogen, halogen, cyano, nitro, trifluoromethyl, OR<sub>5</sub>, SR<sub>5</sub>, NR<sub>5</sub>R<sub>6</sub>, C(O)R<sub>5</sub>, C(O)OR<sub>5</sub>, C(O) NR<sub>5</sub>R<sub>6</sub>, S(O)R<sub>5</sub>, S(O)<sub>2</sub>R<sub>5</sub>, S(O)NR<sub>5</sub>R<sub>6</sub>, S(O)<sub>2</sub>NR<sub>5</sub>R<sub>6</sub>, NR<sub>6</sub>C(O)R<sub>5</sub>, NR<sub>6</sub>C(O)OR<sub>5</sub>, alkyls, alkenyls, alkynyls, aryls, heteroaryls, aralkyls or heteroaralkyls, all optionally substituted; Ra represents in particular halogen, hydroxyl, alkoxy, nitro; Rb represents in particular hydrogen, halogen, cyano, nitro, trifluoromethyle, -W-(C<sub>1</sub>- C<sub>3</sub> alkyl)m- R<sub>5</sub>; R<sub>5</sub> and R<sub>6</sub> represent in particular alkyl, aralkyl or heteroaralkyls optionally substituted; said products being all in the form of isomers and salts, and their use as medicines.</p>
申请公布号 MX2007010278(A) 申请公布日期 2007.11.07
申请号 MX20070010278 申请日期 2006.02.20
申请人 AVENTIS PHARMA S.A. 发明人 JEAN-MARIE RUXER;FABIENNE THOMPSON;PATRICK MAILLIET;LUC BERTIN;CHANTAL CARREZ
分类号 C07D261/20;A61K31/423;A61P35/00 主分类号 C07D261/20
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