发明名称 |
MUSCARINIC RECEPTOR ANTAGONISTS |
摘要 |
Compounds of Formula (I), wherein represents a single bond when G is -OH and double bond when G is -O; R<SUB>1</SUB> and R<SUB>2</SUB> are independently selected from hydrogen, alkyl, alkenyl, alkynyl, aralkyl, cycloalkyl, aryl, heteroaryl, heterocyclyl, heterocyclylalkyl or heteroarylalkyl; R<SUB>3 </SUB>is selected from the group selected from hydrogen, hydroxy, alkoxy, alkenyloxy or alkynyloxy; X is selected from oxygen, -NH, -NR (wherein R is alkyl, alkenyl, alkenyl, alkynyl or aryl), sulphur or no atom; Het is heterocyclyl or heteroaryl; n is an integer from 1 to 6; are muscarinic receptor antagonists, which are useful, among other uses, for the treatment of various diseases of the respiratory, urinary and 4 i gastrointestinal systems mediated through muscarinic receptors. |
申请公布号 |
WO2007077510(A3) |
申请公布日期 |
2007.11.01 |
申请号 |
WO2006IB55010 |
申请日期 |
2006.12.21 |
申请人 |
RANBAXY LABORATORIES LIMITED;KUMAR, NARESH;KAUR, JASKIRAN;PALLE, VENKATA P.;BHATT, BEENU;JINDAL, SHELLY;CHUGH, ANITA;GUPTA, SUMAN;RAY, ABHIJIT;MALHOTRA, SHIVANI;SHIRUMALLA, RAJ KUMAR |
发明人 |
KUMAR, NARESH;KAUR, JASKIRAN;PALLE, VENKATA P.;BHATT, BEENU;JINDAL, SHELLY;CHUGH, ANITA;GUPTA, SUMAN;RAY, ABHIJIT;MALHOTRA, SHIVANI;SHIRUMALLA, RAJ KUMAR |
分类号 |
C07D233/14;A61K31/4164;A61K31/4439;A61P1/00;A61P11/00;A61P13/00;C07D233/60;C07D233/61;C07D401/12 |
主分类号 |
C07D233/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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