发明名称 PROCESSES FOR THE SYNTHESIS OF AZETIDINONE
摘要 Provided are intermediates useful for the synthesis of hydroxyl-alkyl substituted azetidinones, processes of their preparation, and processes for the synthesis of certain hydroxyl-alkyl substituted azetidinones. Also provided are processes for the synthesis ofl-(4-fluorophenyl)-3(R)-[3-(4-fluorophenyl)-3(S)- hydroxypropyl]-4(S)-(4-hydroxyphenyl)-2-azetidinone, or ezetimibe.
申请公布号 WO2007120824(A2) 申请公布日期 2007.10.25
申请号 WO2007US09132 申请日期 2007.04.10
申请人 TEVA PHARMACEUTICAL INDUSTRIES LTD.;TEVA PHARMACEUTICALS USA, INC.;KANSAL, KINOD, KUMAR;AHMAD, SUHAIL;MARIAPPAN, SHANMUGAVEL;TYAGI, BHUPENDRA;PERLMAN, NURIT;LE PAIH, JACQUES;ZANOTTI-GEROSA, ANTONIO 发明人 KANSAL, KINOD, KUMAR;AHMAD, SUHAIL;MARIAPPAN, SHANMUGAVEL;TYAGI, BHUPENDRA;PERLMAN, NURIT;LE PAIH, JACQUES;ZANOTTI-GEROSA, ANTONIO
分类号 C07D413/06;C07D405/06;C07D417/06 主分类号 C07D413/06
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