发明名称 |
PROCESSES FOR THE PREPARATION OF 8-CHLORO-1-METHYL-2,3,4,5-TETRAHYDRO-1H-3-BENZAZEPINE AND INTERMEDIATES RELATED THERETO |
摘要 |
The present invention provides processes, methods and intermediates for the preparation of 8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine, salts, hydrates and crystal forms thereof which are useful as serotonin (5-HT) receptor agonists for the treatment of, for example, central nervous system disorders such as obesity. |
申请公布号 |
WO2007120517(A2) |
申请公布日期 |
2007.10.25 |
申请号 |
WO2007US08170 |
申请日期 |
2007.04.02 |
申请人 |
ARENA PHARMACEUTICALS, INC.;WEIGL, ULRICH;PORSTMANN, FRANK;STRAESSLER, CHRISTOPH;ULMER, LARS;KOETZ, ULF |
发明人 |
WEIGL, ULRICH;PORSTMANN, FRANK;STRAESSLER, CHRISTOPH;ULMER, LARS;KOETZ, ULF |
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