发明名称 |
AZOLYLACYLGUANIDINES AS beta;-SECRETASE INHIBITORS |
摘要 |
The present invention provides an azolylacylquanidine compound of formula (I). The present invention also provides methods for the use thereof to inhibit F-secretase (BACE) and treat F-amyloid deposits and neurofibrillary tangles.
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申请公布号 |
KR20070102751(A) |
申请公布日期 |
2007.10.19 |
申请号 |
KR20077020831 |
申请日期 |
2007.09.11 |
申请人 |
WYETH |
发明人 |
COLE DEREK CECIL;MANAS ERIC STEVEN;JENNINGS LEE DALTON;LOVERING FRANK ELDRIDGE;STOCK JOSEPH RAYMOND;MOORE WILLIAM JAY;ELLINGBOE JOHN WATSON;CONDON JEFFREY SCOTT;SUKHDEO MOHANI NIRMALA;ZHOU PING;WU JUNJUN;MORRIS KOI MICHELE |
分类号 |
C07D207/327;C07D207/32;C07D409/04;C07D413/04 |
主分类号 |
C07D207/327 |
代理机构 |
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