发明名称 METHOD FOR PRODUCING TETRAHYDRO-PYRIDOAZEPIN-8-ONE COMPOUND
摘要 PROBLEM TO BE SOLVED: To provide a method for producing a tetrahydro-pyridoazepin-8-one compound. SOLUTION: The method for producing the 2-ä4-[4-(7-fluoronaphthalen-1-yl)-piperazin-1-yl]butoxy}-5,6,7,9-tetrahydro-1,7,9-triaza-benzocyclohepten-8-one comprises reacting 1-(7-fluoronaphthalen-1-yl)-piperazine hydrochloride with a compound represented by formula (II) äwherein, L is a leaving group}. COPYRIGHT: (C)2008,JPO&INPIT
申请公布号 JP2007269796(A) 申请公布日期 2007.10.18
申请号 JP20070090495 申请日期 2007.03.30
申请人 PFIZER PROD INC 发明人 CHEN MICHAEL HUAI GU;MAGANO JAVIER;MENNEN KENNETH EARL
分类号 C07D471/04;A61K31/5513;A61P25/00 主分类号 C07D471/04
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