发明名称 ПИРРОЛОПИРИМИДИНОНОВЫЕ ПРОИЗВОДНЫЕ
摘要 A compound having GSK-3 inhibitory activity. A 1 and A 3 are a single bond, an aliphatic hydrocarbon; A 2 and A 4 are a single bond, CO, COO, etc.; G 1 is a single bond, an alicyclic hydrocarbon, aromatic hydrocarbon, etc.; G 2 is H, an aliphatic hydrocarbon, an alicyclic hydrocarbon, an aromatic hydrocarbon, etc.; A 5 is a single bond, NR; R 2 is H, halogen, an aliphatic hydrocarbon, etc.; A 6 is a single bond, NR, CO, etc.; R 3 is H, halogen, nitro, saturated aliphatic hydrocarbon, etc.; and wherein R is H or an lower aliphatic hydrocarbon group.
申请公布号 RU2006109503(A) 申请公布日期 2007.10.10
申请号 RU20060109503 申请日期 2004.08.26
申请人 ТЕЙДЗИН ФАРМА ЛИМИТЕД (JP) 发明人 ЦУЦУМИ Такахару (JP);СУГИУРА Сатоси (JP);КОГА Масахиро (JP);МАЦУМОТО Есиюки (JP);ИСИИ Тосихиро (JP);НАКАНО Акира (JP);УНОКИ Ген (JP);САКАИ Юри (JP);ТАКАРАДА Рейко (JP);ОГАВА Хироко (JP)
分类号 C07D487/04;A61K31/519;A61P3/10;A61P17/14;A61P25/24;A61P25/28;A61P29/00;A61P35/00;A61P37/02;A61P43/00;C07D487/02 主分类号 C07D487/04
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