发明名称 Compounds useful as reversible inhibitors of cysteine proteases
摘要 Disclosed are novel cathepsin S, K, F, L and B reversible inhibitory compounds of the formulas (I), (II), (Ia) and (Ib) further defined herein. The compounds are useful for treating autoimmune diseases. Also disclosed are processes for making such novel compounds
申请公布号 US7279472(B2) 申请公布日期 2007.10.09
申请号 US20040937636 申请日期 2004.09.09
申请人 BOEHRINGER INGELHEIM PHARMACEUTICALS INC. 发明人 EMMANUEL MICHEL JOSE;FRYE LEAH L.;HICKEY EUGENE R.;LIU WEIMIN;MORWICK TINA MARIE;SPERO DENICE MARY;SUN SANXING;THOMSON DAVID S.;WARD YANCEY DAVID;YOUNG ERICK RICHARD ROUSH
分类号 A61K31/535;A61K31/40;A61K31/4468;A61K31/454;A61K31/496;A61K31/497;A61K31/506;A61K31/517;A61K31/5365;A61K31/5377;A61K31/538;A61K31/541;A61K31/55;A61P1/04;A61P3/10;A61P9/10;A61P11/06;A61P19/10;A61P21/04;A61P25/28;A61P29/00;A61P31/00;A61P37/00;A61P37/06;C07D205/04;C07D207/14;C07D207/16;C07D211/58;C07D211/60;C07D211/66;C07D309/14;C07D335/02;C07D401/04;C07D401/12;C07D403/06;C07D405/12;C07D413/02;C07D413/12;C07D413/14;C07D417/12;C07D455/02;C07D487/08 主分类号 A61K31/535
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