发明名称 |
4- (2, 6-DICHLOROBENZOYLAMINO) -lH-PYRAZOLE-3 -CARBOXYLIC ACID PIPERIDIN- 4 -YLAMID ACID ADDITION SALTS AS KINASE INHIBITORS. |
摘要 |
<p>The invention provides an acid addition salt of 4-(2,6-dichloro-benzoylamino)-lH- pyrazole-3-carboxylic acid piperidin-4-ylamide and crystals thereof, the salt being formed with an acid selected from methanesulphonic acid and acetic acid and mixtures thereof. Also provided are the novel uses of salts of 4-(2,6-dichloro-benzoylamino)-lH- pyrazole-3-carboxylic acid piperidin-4-ylamide, processes for the preparation of 4- (2,6-dichloro-benzoylamino)-lH-pyrazole-3-carboxylic acid piperidin-4-ylamide and its salts and novel chemical intermediates.</p> |
申请公布号 |
MX2007008783(A) |
申请公布日期 |
2007.09.11 |
申请号 |
MX20070008783 |
申请日期 |
2006.01.20 |
申请人 |
ASTEX THERAPEUTICS LIMITED |
发明人 |
GARY TREWARTHA;PAUL GRAHAM WYATT;DAVID CHARLES REES;MLADEN VINKOVIC |
分类号 |
C07D401/12;A61K31/4155;A61K31/454;A61P35/00;A61P35/02 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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