| 摘要 |
8-Substituted-2,6-methano-3-benzazocines of general structure I in which A is -CH<SUB>2</SUB>-OH, -CH<SUB>2</SUB>NH<SUB>2</SUB>, -NHSO<SUB>2</SUB>CH<SUB>3</SUB>, and Y is O, S or NOH are useful as analgesics, anti-diarrheal agents, anticonvulsants, antitussives and anti-addiction medications. 8-Carboxamides, thiocarboxamides, hydroxyamidines and formamides are preferred.
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