发明名称 |
CRYSTALLINE FORMS OF (3R,4R)-4-AMINO-1-[[4-[(3-METHOXYPHENYL)AMINO]PYRROLO[2,1-F][1,2,4]TRIAZIN-5-YL]METHOL]PIPERIDIN-3-OL |
摘要 |
<p>Crystalline forms of (3R,4R)-4-amino-1-[[4-[(3-methoxyphenyl)amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]piperidin-3-ol of the formula (I) are provided. Also provided is a pharmaceutical composition comprising one or more crystalline forms of (3R,4R)-4-amino-1-[[4-[(3-methoxyphenyl)amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]piperidin-3-ol, as well as a method of using one or more crystalline forms of (3R,4R)-4-amino-1-[[4-[(3-methoxyphenyl)amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]piperidin-3-ol in the treatment of cancer and other proliferative diseases.</p> |
申请公布号 |
WO2007095632(A1) |
申请公布日期 |
2007.08.23 |
申请号 |
WO2007US62276 |
申请日期 |
2007.02.16 |
申请人 |
BRISTOL-MYERS SQUIBB COMPANY;WEI, CHENKOU;NORRIS, DEREK, J. |
发明人 |
WEI, CHENKOU;NORRIS, DEREK, J. |
分类号 |
C07D487/04;A61K31/53;A61P35/00 |
主分类号 |
C07D487/04 |
代理机构 |
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主权项 |
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地址 |
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