发明名称 |
N-substituted nonaryl-heterocyclo amidyl NMDA/NR2B Antagonists |
摘要 |
Compounds represented by Formula (I): or pharmaceutically acceptable salts thereof, are effective as NMDA NR2B antagonists useful for relieving pain.
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申请公布号 |
US7259157(B2) |
申请公布日期 |
2007.08.21 |
申请号 |
US20020114685 |
申请日期 |
2002.04.02 |
申请人 |
MERCK & CO., INC. |
发明人 |
LIVERTON NIGEL J.;BUTCHER JOHN W.;MCINTYRE CHARLES;CLAIBORNE CHRISTOPHER F.;CLAREMON DAVID A.;MCCAULEY JOHN A.;ROMANO JOSEPH J.;THOMPSON WAYNE;MUNSON PETER M. |
分类号 |
A61K31/554;A61K31/40;A61K31/425;A61K31/44;A61K31/445;A61K31/451;A61K31/4535;A61K31/454;A61K31/4545;A61K31/4709;A61K31/4725;A61K31/495;A61K31/496;A61K31/4965;A61K31/497;A61K31/501;A61K31/506;A61K31/519;A61K31/52;A61K31/5375;A61K31/5377;A61K31/55;A61K31/553;A61P9/10;A61P25/04;A61P25/06;A61P25/16;A61P25/18;A61P25/22;A61P25/24;A61P27/06;A61P27/16;C07D207/09;C07D211/26;C07D211/38;C07D211/42;C07D211/96;C07D241/04;C07D265/30;C07D267/10;C07D401/12;C07D401/14;C07D405/14;C07D409/12;C07D409/14;C07D413/12;C07D417/04;C07D417/12;C07D417/14;C07D471/04;C07D473/00;C07D487/04 |
主分类号 |
A61K31/554 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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