发明名称 CRYSTALLINE FORMS OF (3R,4R)-4-AMINO-1-[[4-[(3-METHOXYPHENYL)AMINO]PYRROLO[2,1-f][1,2,4]TRIAZIN-5-YL]METHYL]PIPERIDIN-3-OL
摘要 Crystalline forms of (3R,4R)-4-amino-1-[[4-[(3-methoxyphenyl)amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]piperidin-3-ol of the formula are provided. Also provided is a pharmaceutical composition comprising one or more crystalline forms of (3R,4R)-4-amino-1-[[4-[(3-methoxyphenyl)amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]piperidin-3-ol, as well as a method of using one or more crystalline forms of (3R,4R)-4-amino-1-[[4-[(3-methoxyphenyl)amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]methyl]piperidin-3-ol in the treatment of cancer and other proliferative diseases.
申请公布号 US2007191375(A1) 申请公布日期 2007.08.16
申请号 US20070675108 申请日期 2007.02.15
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 WEI CHENKOU;NORRIS DEREK J.
分类号 A61K31/53;C07D487/04 主分类号 A61K31/53
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