发明名称 Novel compounds that are ERK inhibitors
摘要 Disclosed are the ERK inhibitors of formula 1.0: and the pharmaceutically acceptable salts and solvates thereof. Q is a piperidine or piperazine ring that can have a bridge or a fused ring. The piperidine ring can have a double bond in the ring. All other substitutents are as defined herein. Also disclosed are methods of treating cancer using the compounds of formula 1.0.
申请公布号 US2007191604(A1) 申请公布日期 2007.08.16
申请号 US20060636954 申请日期 2006.12.11
申请人 COOPER ALAN;DENG YONGQI;SHIPPS GERALD W JR;SHIH NENG-YANG;ZHU HUGH;SUN ROBERT;KELLY JOSEPH M;DOLL RONALD;NAN YANG;WANG TONG;DESAI JAGDISH;WANG JAMES J;DONG YOUHAO;MADISON VINCENT;XIAO LI;HRUZA ALAN W;SIDDIQUI M A;SAMATAR AHMED A;PALIWAL SUNIL;TSUI HON-CHUNG;CELEBI AZIM A;WU YIJI;BOGA SOBHANA B 发明人 COOPER ALAN;DENG YONGQI;SHIPPS GERALD W.JR.;SHIH NENG-YANG;ZHU HUGH;SUN ROBERT;KELLY JOSEPH M.;DOLL RONALD;NAN YANG;WANG TONG;DESAI JAGDISH;WANG JAMES J.;DONG YOUHAO;MADISON VINCENT;XIAO LI;HRUZA ALAN W.;SIDDIQUI M. A.;SAMATAR AHMED A.;PALIWAL SUNIL;TSUI HON-CHUNG;CELEBI AZIM A.;WU YIJI;BOGA SOBHANA B.
分类号 C07D417/14;C07D403/14;C07D413/14 主分类号 C07D417/14
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