发明名称 |
Multicore indazolinone library |
摘要 |
There is provided a method to convert O-functionalized indazolinone-derivatives to the corresponding N2-functionalized indazolinone derivatives, by use of microwave energy or a transition metal catalyst. A preferred catalyst is palladium tetrakis. The method described allows the creation of a library of chemical compounds which can be screened for biological activity.
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申请公布号 |
US2007179294(A1) |
申请公布日期 |
2007.08.02 |
申请号 |
US20050629150 |
申请日期 |
2005.06.08 |
申请人 |
THE UNIVERSITY COURT OF THE UNIVERSITY OF ST ANDREWS |
发明人 |
WESTWOOD NICHOLAS J.;ISAMBERT NICHOLAS S.J. |
分类号 |
C07D475/00;C07D231/00;C07D231/56 |
主分类号 |
C07D475/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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