发明名称 FUSED AZEPINE DERIVATIVES AND THEIR USE AS ANTIDIURETIC AGENTS
摘要 Compounds according to general formulae (1 and 2), wherein G<SUP>1 </SUP>is an azepine derivative and G<SUP>2 </SUP>is a group according to general formulae (9-11) are new. Compounds according to the invention are vasopressin V<SUB>2 </SUB>receptor agonists. Pharmaceutical compositions of the compounds are useful as antidiuretic agents
申请公布号 EP1294698(B1) 申请公布日期 2007.08.01
申请号 EP20010940792 申请日期 2001.06.21
申请人 FERRING B.V. 发明人 ASHWORTH, DOREEN MARY;PITT, GARY ROBERT WILLIAM;HUDSON, PETER;YEA, CHRISTOPHER MARTYN;FRANKLIN, RICHARD JEREMY;SEMPLE, GRAEME;JENKINS, PAUL DAVID
分类号 C07D223/16;A61K31/55;A61K31/551;A61K31/5513;A61K31/5517;A61K31/553;A61K31/554;A61P13/00;A61P13/02;A61P25/00;A61P43/00;C07D243/12;C07D243/14;C07D255/04;C07D267/14;C07D281/10;C07D401/06;C07D401/12;C07D403/12;C07D413/12;C07D471/04;C07D487/04;C07D495/04;C07D498/04;C07D519/00 主分类号 C07D223/16
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