DNT-BENZENESULFONATE AND METHODS OF PREPARATION THEREOF
摘要
<p>(S)-N,N-Dimethyl-3-(l-naphthalenyloxy)-3-(2-thienyl)propanamine benzenesulfonate (DNT-benzenesulfonate) and polymorphs of DNT-benzenesulfonate, compositions of DNT-benzenesulfonate and its polymorphs, processes for the preparation of DNT-benzenesulfonate and its polymorphs, and processes for the preparation of duloxetine hydrochloride from DNT-benzenesulfonate are provided.</p>
申请公布号
WO2007084194(A1)
申请公布日期
2007.07.26
申请号
WO2006US36976
申请日期
2006.09.21
申请人
TEVA PHARMACEUTICAL INDUSTRIES LTD.;TEVA PHARMACEUTICALS USA, INC.;INI, SANTIAGO;ABRAMOV, MILI;KOLTAI, TAMAS