发明名称 Resolution of 3-amino alkylnitriles
摘要 The present invention relates to chiral N-acetyl-alpha-amino acid salts of optically active beta-amino alkylnitriles, and also to a process for preparing optically active beta-amino alkylnitriles by resolving racemic beta-amino alkylnitriles using chiral N-acetyl-alpha-amino acids as resolving agent.
申请公布号 ZA200603356(B) 申请公布日期 2007.07.25
申请号 ZA20060003356 申请日期 2006.04.24
申请人 PFIZER PRODUCTS INC. 发明人 COLBERG, JUAN CARLOS;MOTTERLE, RICCARDO;ZAMBELLI FRANZ, SAMUELA;STIVANELLO, MARIANO
分类号 A61K31/277;A61K31/401;A61K31/405;A61K31/4172;C07B;C07B57/00;C07C;C07C253/32;C07C255/24;C07C255/29;C07D233/90 主分类号 A61K31/277
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