发明名称 PYRROLOPYRIMIDINE AND PYRROLOPYRIDINE DERIVATIVE SUBSTITUTED WITH CYCLIC AMINO GROUP
摘要 PROBLEM TO BE SOLVED: To provide a CRF receptor antagonist and/or aδ-receptor agonist which are effective as a medicine for treating or preventing diseases considered to participate in CRF, such as depression, anxiety, Alzheimer's disease, Parkinson's disease, Huntington's chorea, feeding disorders, hypertension, gastrointestinal disease, drug dependency, cerebral infarction, cerebral ischemia, cerebral edema, head trauma, inflammation, immiity-related diseases, alopecia, irritable intestine syndromes, somnipathy, epilepsy, dermatitis, integrated ataxia, and ache. SOLUTION: The pyrrolopyrimidine or pyrrolopyridine derivative substituted with a cyclic amino group, represented by formula [I], has high affinity with the CRF receptor and/or theδ-receptor, and is effective for diseases estimated to participate in CRF. COPYRIGHT: (C)2007,JPO&INPIT
申请公布号 JP2007169216(A) 申请公布日期 2007.07.05
申请号 JP20050369410 申请日期 2005.12.22
申请人 TAISHO PHARMACEUT CO LTD 发明人 NAKAZATO ATSUO;OKUBO TAKETOSHI;NOZAWA MASARU;TAMIDA TOMOKO;KENNIS LUDO E J
分类号 A61K31/4545;A61K31/519;A61K31/662;A61P1/00;A61P9/10;A61P9/12;A61P17/00;A61P17/14;A61P25/00;A61P25/04;A61P25/08;A61P25/16;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P29/00;A61P37/00;C07D471/04;C07D487/04;C07D519/00 主分类号 A61K31/4545
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