发明名称 BENZOAZOLYPIPERAZINE DERIVATIVES HAVING VR1 ANTAGONISTIC ACTIVITY
摘要 A compound of formula: wherein Ar1, A, R3, X, and m are as disclosed herein and Ar2 is a benzothiazolyl, benzooxazolyl, or benzoimidazolyl group or a pharmaceutically acceptable salt thereof (a “Benzoazolylpiperazine Compound”), compositions comprising a Benzoazolylpiperazine Compound, and methods for treating or preventing pain, UI, an ulcer, IBD, IBS, an addictive disorder, Parkinson's disease, parkinsonism, anxiety, epilepsy, stroke, a seizure, a pruritic condition, psychosis, a cognitive disorder, a memory deficit, restricted brain function, Huntington's chorea, amyotrophic lateral sclerosis, dementia, retinopathy, a muscle spasm, a migraine, vomiting, dyskinesia, or depression in an animal comprising administering to an animal in need thereof an effective amount of a Benzoazolylpiperazine Compound are disclosed.
申请公布号 IL169378(D0) 申请公布日期 2007.07.04
申请号 IL20050169378 申请日期 2005.06.23
申请人 EURO-CELTIQUE S.A 发明人
分类号 A61K31/495;A61K31/496;A61P13/00;A61P29/00;C07D;C07D401/12;C07D403/12;C07D413/12;C07D417/12;C07D417/14 主分类号 A61K31/495
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