发明名称 |
Heterocycles and uses thereof |
摘要 |
Compounds of the following formula are disclosed: wherein R<SUP>B </SUP>is a substituted or unsubstituted aryl or heteroaryl moiety; at least one of R<SUP>U </SUP>and R<SUP>L </SUP>is a phosphorus-containing moiety, J, and the other of R<SUP>U </SUP>and R<SUP>L </SUP>is independently chosen from H; halogen; -CN; -NO<SUB>2</SUB>; -J; -SO<SUB>2</SUB>R; -SO<SUB>2</SUB>NRR'; or -ZR<SUP>J</SUP>, wherein each occurrence of Z is independently -O-, -S- or -NR- and each occurrence of R<SUP>J </SUP>is independently -R, -COR, -COOR or -CONRR'.
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申请公布号 |
US7238679(B2) |
申请公布日期 |
2007.07.03 |
申请号 |
US20030744601 |
申请日期 |
2003.12.23 |
申请人 |
ARIAD PHARMACEUTICALS, INC. |
发明人 |
KEENAN TERENCE P.;SHAKESPEARE WILLIAM C. |
分类号 |
A61K31/517;A01N57/00;A61K31/675;C07D211/32;C07D233/00;C07D249/04;C07D257/10;C07D263/30;C07D277/20;C07D403/00;C07D413/00;C07F9/02;C07F9/6512;C07F9/6558 |
主分类号 |
A61K31/517 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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