发明名称 PROCESS TO PREPARE SUBSTITUTED IMIDAZOPYRAZINE COMPOUNDS
摘要 <p>A method of preparing formula (A) ,wherein, X=C1, Br, I, comprises the step of treating formula (B), with N-chloro-, N-bromo-, or N-iodosuccinimide in a compatible solvent such as dimethylformamide (DMF) at 0-60° C followed by halogenation.</p>
申请公布号 WO2007067709(A1) 申请公布日期 2007.06.14
申请号 WO2006US46764 申请日期 2006.12.07
申请人 OSI PHARMACEUTICALS, INC.;MULVIHILL, KRISTEN, MICHELLE;CASTELHANO, ARLINDO, L. 发明人 MULVIHILL, KRISTEN, MICHELLE;CASTELHANO, ARLINDO, L.
分类号 C07D487/04 主分类号 C07D487/04
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