| 发明名称 |
SOMATOSTATIN RECEPTOR ANTAGONIST |
| 摘要 |
<p><P>PROBLEM TO BE SOLVED: To provide a new somatostatin receptor (SSTR) antagonist and a medicine using the same as an active ingredient. <P>SOLUTION: This somatostatin receptor antagonist is expressed by: Cpa-cyclo(D-Cys-4-Pal-D-Trp-Lys-Thr-Cys)-Nal-NH<SB>2</SB>or its pharmaceutically acceptable salt. The use of the compound as the somatostatin receptor antagonist is provided. The medicinal composition containing the compound and having the somatostatin receptor antagonist activity is also provided. The composition is anticipated to have the treating effect of medullary thyroid cancer. <P>COPYRIGHT: (C)2007,JPO&INPIT</p> |
| 申请公布号 |
JP2007145854(A) |
申请公布日期 |
2007.06.14 |
| 申请号 |
JP20070005725 |
申请日期 |
2007.01.15 |
| 申请人 |
IL CONSORZIO FERRARA RICHERCHE;SOC DE CONSEILS DE RECHERCHES & D'APPLICATIONS SCIENTIFIQUES SAS |
发明人 |
DEGLI UBERTI ETTORE CIRO;ZATELLI MARIA CHIARA;CULLER MICHAEL DEWITT |
| 分类号 |
C07K7/54;G01N33/48;A61K38/00;A61K38/08;A61K38/31;A61K45/00;A61K51/00;A61P5/02;A61P35/00;A61P35/04;A61P43/00;C07K7/06;C07K7/64;C12N5/06;C12Q1/02;G01N33/68 |
主分类号 |
C07K7/54 |
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