发明名称 3-AMINO-2-ARYLPROPYL AZAINDOLES AND USES THEREOF
摘要 <p>The present invention provides compounds of the formula I: or pharmaceutically acceptable salts, solvates or prodrugs thereof, wherein p, Ar, R&lt;SUP&gt;1&lt;/SUP&gt;, R&lt;SUP&gt;2&lt;/SUP&gt;, R&lt;SUP&gt;3&lt;/SUP&gt;, R&lt;SUP&gt;a&lt;/SUP&gt;, R&lt;SUP&gt;b&lt;/SUP&gt;, R&lt;SUP&gt;c&lt;/SUP&gt;, R&lt;SUP&gt;d&lt;/SUP&gt; and R&lt;SUP&gt;e&lt;/SUP&gt; are defined herein. Also provided are pharmaceutical compositions, methods of using, and methods of preparing the compounds. The compounds are useful for the treatment of diseases associated with monoamine reuptake inhibitors.</p>
申请公布号 WO2007062998(A1) 申请公布日期 2007.06.07
申请号 WO2006EP68650 申请日期 2006.11.20
申请人 F. HOFFMANN-LA ROCHE AG;GREENHOUSE, ROBERT;JAIME-FIGUEROA, SAUL;LYNCH, STEPHEN M.;RAPTOVA, LUBICA;STEIN, KARIN ANN;WEIKERT, ROBERT JAMES 发明人 GREENHOUSE, ROBERT;JAIME-FIGUEROA, SAUL;LYNCH, STEPHEN M.;RAPTOVA, LUBICA;STEIN, KARIN ANN;WEIKERT, ROBERT JAMES
分类号 C07D471/04;A61K31/395;A61K31/437;A61P25/22;A61P25/24;C07D487/04;C07D487/14 主分类号 C07D471/04
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