发明名称 BENZOAZOLYPIPERAZINE DERIVATIVES HAVING VR1 ANTAGONISTIC ACTIVITY
摘要 A compound of formula (I) wherein Ar1, A, R3, x, and m are as disclosed herein and Ar2 is a benzothiazolyl, benzooxazolyl, or benzoimidazolyl group or a pharmaceutically acceptable salt thereof (Benzoazolylpiperazine Compound), compositions comprising a Benzoazolylpiperazine Compound, and methods for treating or preventing pain, UI, an ulcer, IBD, IBS, an addictive disorder, Parkinson disease, parkinsonism, anxiety, epilepsy, stroke, a seizure, a pruritic condition, psychosis, a cognitive disorder, a memory deficit, retricted brain function, Huntington- chorea, amyotrophic lateral sclerosis, dementia, retinopathy, a muscle spasm, a migraine, vomiting, dyskinesia, or depression in an animal comprising administering to an animal in need thereof an effective amount of Benzoazolylpiperazine Compound are disclosed.
申请公布号 RS20050498(A) 申请公布日期 2007.06.04
申请号 YU2005P000498 申请日期 2003.12.22
申请人 EUROCELTIQUE S.A. 发明人 SUN QUN;TAFESSE LAYKEA;VICTORY SAM
分类号 C07D417/12;A61K31/495;A61K31/496;A61P13/00;A61P29/00;C07D401/12;C07D403/12;C07D413/12;C07D417/14 主分类号 C07D417/12
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