发明名称 NOVEL METHOD OF PREPARATION OF 5-CHLORO-3-IMIDAZOL-1-YL-[1,2,4]THIADIAZOLE AND (3-IMIDAZOL-1-YL-[1,2,4]THIADIAZOL-5YL)-DIALKYL-AMINES
摘要 The present invention discloses a novel method for preparing 3-imidazol-1-yl-[1,2,4]thiadiazole derivatives, particularly to a method of preparing 5-halo-3-imidazol-1-yl-[1,2,4]thiadiazole, more particularly (3 -imidazol-1-yl-[1,2,4]thiadiazol-5-yl)-dialkyl-amines, that afford a high yield of pure product.
申请公布号 US2007123572(A1) 申请公布日期 2007.05.31
申请号 US20060563200 申请日期 2006.11.25
申请人 KALYPSYS, INC. 发明人 HERBERT MARK R.;COUSINS RUSSELL D.;LANG HENGYUAN;GAHMAN TIMOTHY C.;NOBLE STEWART A.
分类号 A61K31/433;C07D417/04 主分类号 A61K31/433
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