发明名称 |
METHODS FOR PRODUCING ISOINDOLE DERIVATIVES |
摘要 |
The present invention relates to a method for producing an isoindole derivative (compound (II)) with the following general formula (II):
(wherein R 1 and R 2 each independently represents a C 1-6 alkyl group) or a salt thereof, comprising the step of cyclizing, in a solvent, compound (I) with the following general formula (I):
(wherein R 1 and R 2 have the same meanings as R 1 and R 2 in formula (II) above) or a salt thereof, or their hydrate or solvate in the presence of a base (Step 1).
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申请公布号 |
EP1787983(A1) |
申请公布日期 |
2007.05.23 |
申请号 |
EP20050766977 |
申请日期 |
2005.07.27 |
申请人 |
EISAI R&D MANAGEMENT CO., LTD. |
发明人 |
YOSHIZAWA, KAZUHIRO;NAKAMURA, TAIJU;NEGI, SHIGETO |
分类号 |
C07D209/44;C07C255/59 |
主分类号 |
C07D209/44 |
代理机构 |
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代理人 |
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地址 |
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